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Meta-Cyanobenzyl substituted benzimidazolium salts: Synthesis, characterization, crystal structure and carbonic anhydrase, -glycosidase, butyrylcholinesterase, and acetylcholinesterase inhibitory properties
(Wiley, 2018-07)
meta-Cyanobenzyl-substituted N-heterocyclic carbene (NHC) precursors were synthesized by the reaction of a series of N-(alkyl)benzimidazolium with 3-bromomethyl-benzonitrile. These benzimidazolium salts were characterized ...
Synthesis of chalcone-imide derivatives and investigation of their anticancer and antimicrobial activities, carbonic anhydrase and acetylcholinesterase enzymes inhibition profiles
(Taylor & Francis, 2018)
The new 1-(4-(3-(aryl)acryloyl)phenyl)-1H-pyrrole-2,5-diones (5a-g) were prepared from 4-aminchalcones (3a-g) and screened for biological activities. All compounds (3a-g and 5a-g), except 3d and 3e displayed good cytotoxic ...
The impact of some natural phenolic compounds on carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase, and -glycosidase enzymes: An antidiabetic, anticholinergic, and antiepileptic study
(Wiley, 2017-12)
Natural products from food and plant sources have been used for medicinal usage for ages. Also, natural products with therapeutic significance are compounds derived from animals, plants, or any microorganism. In this study, ...
Synephrine and phenylephrine act as -amylase, -glycosidase, acetylcholinesterase, butyrylcholinesterase, and carbonic anhydrase enzymes inhibitors
(Wiley, 2017-11)
In this paper, synephrine and phenylephrine compounds showed excellent inhibitory effects against human carbonic anhydrase (hCA) isoforms I and II, -amylase, -glycosidase, acetylcholinesterase (AChE), and butyrylcholinesterase ...
Synthesis and investigation of anticancer, antibacterial activities and carbonic anhydrase, acetylcholinesterase inhibition profiles of novel (3aR,4S,7R,7aS)-2-[4-[1-acetyl-5-(aryl/heteroaryl)-4,5-dihydro-1H-pyrazol-3-yl]phenyl]-3a,4,7,7a-tetrahydro-1H-4,7-methanoisoindole-1,3(2H)-diones
(MONATSHEFTE FUR CHEMIE, 2019-04)
A series of novel 1,3,5-trisubstituted pyrazoline derivatives, (3aR,4S,7R,7aS)-2-[4-[1-acetyl-5-(aryl/heteroaryl)-4,5-dihydro-1H-pyrazol-3-yl]phenyl]-3a,4,7,7a-tetrahydro-1H-4,7-methanoisoindole-1,3(2H)-diones, were ...
Sosyal bilgiler dersi ve kültür aktarımında edindiği rol üzerine bir inceleme
(Yeni Eğitim Yayıncılık, 2019)
Bu çalışmada, sosyal bilgiler dersi ve bu dersin kültür aktarımında üstlendiği rolün incelenmesi amaçlanmıştır. Bu kapsamda öncelikle sosyal bilgiler dersinin tarihi gelişimi, nasıl bir doğaya sahip olduğu, kültür kavramı ...
Some pyrazoles derivatives: Potent carbonic anhydrase, α‐glycosidase, and cholinesterase enzymes inhibitors
(Wiley, 2018-10)
A series of substituteed pyrazol-4-yl-diazene derivatives were found to be effective inhibitors against -glycosidase, cytosolic carbonic anhydrase I and II isoforms (hCA I and II), butyrylcholinesterase (BChE), and ...
Inhibitory effects of oxytocin and oxytocin receptor antagonist atosiban on the activities of carbonic anhydrase and acetylcholinesterase enzymes in the liver and kidney tissues of rats
(Wiley, 2017-11)
The aim of this study was to investigate the effects of oxytocin (OT), atosiban, which is an OT receptor antagonist, and OT-atosiban chemicals injected to rats on the activities of carbonic anhydrase (CA) and acetylcholinesterase ...
Sınıf ve sosyal bilgiler öğretmenlerinin ilkokul 4. sınıf insan hakları, yurttaşlık ve demokrasi dersine yönelik görüşlerinin karşılıklı olarak incelenmesi
(Ahi Evran Üniversitesi Kırşehir Üniversitesi Eğitim Fakütlesi, 2016)
Eğitim bireyin davranışlarında istenilen yönde değişim gerçekleştirmeyi amaçlar. Bunu yaparken bireyi kişisel, sosyal, ekonomik ve siyasi alanlarda gerekli bilgi ve donanıma sahip olarak yetiştirmeyi de hedefler. Bu ...
Sosyal bilgiler dersinde değer aktarımı açısından Sadî Şirazî’nin “Bostan” ve “Gülistan” isimli eserlerinin incelenmesi
(Erzin Üniversitesi Eğitim Fakütlesi, 2016)
Değerlerin uygun bir eğitim anlayışı ile bireylere aktarımı konusunda farklı modeller üzerinde durulmaktadır. Bunlardan birisi de edebi eserlerin kullanımıdır. Bu araştırmada, sosyal bilgiler dersi kapsamında değer aktarımı ...