Browsing Fen Fakültesi by Author "Yakup, Budak"

Now showing items 1-2 of 2

Synthesis and investigation of antibacterial activities and carbonic anhydrase and acetyl cholinesterase inhibition profiles of novel 4,5-dihydropyrazol and pyrazolyl-thiazole derivatives containing methanoisoindol-1,3-dion unit

Yakup, Budak; Umit M., Kocyigit; Meliha Burcu, Gurdere; Kezban, Ozcan; Parham, Taslimi; Ilhami, Gulcin; Mustafa, Ceylan (Taylor & Francis, 2017)

Novel 4,5-dihydropyrazole derivatives (3a-i), 3-(4-((3aR,4S,7R,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydro-1H-4,7-methanoisoindol-2(3H)-yl)phenyl)-5-phenyl-4,5-dihydro-1H-pyrazole-1-carbothio amide, were obtained by the addition ...
Synthesis of chalcone-imide derivatives and investigation of their anticancer and antimicrobial activities, carbonic anhydrase and acetylcholinesterase enzymes inhibition profiles

Umit Muhammet, Kocyigit; Yakup, Budak; Meliha Burcu, Gurdere; Fatih, Erturk; Belkiz, Yencilek; Taslimi, Parham; Ilhami, Gulcin; Mustafa, Ceylan (Taylor & Francis, 2018)

The new 1-(4-(3-(aryl)acryloyl)phenyl)-1H-pyrrole-2,5-diones (5a-g) were prepared from 4-aminchalcones (3a-g) and screened for biological activities. All compounds (3a-g and 5a-g), except 3d and 3e displayed good cytotoxic ...