Ara
Toplam kayıt 249, listelenen: 61-70
Discovery of potent carbonic anhydrase, acetylcholinesterase, and butyrylcholinesterase enzymes inhibitors: The new amides and thiazolidine-4-ones synthesized on an acetophenone base
(Wiley, 2017-09)
Compounds containing nitrogen and sulfur atoms can be widely used in various fields, including industry, medicine, biotechnology, and chemical technology. Among them, amides of acids and heterocyclic compounds have an ...
Synthesis, carbonic anhydrase I and II inhibition studies of the 1,3,5-trisubstituted-pyrazolines
(Informa, 2017)
4-(3-(4-Substituted-phenyl)-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl) benzenesulfonamides (9-16) were successfully synthesized and their chemical structures were confirmed by H-1 NMR, C-13 NMR, and HRMS spectra. Carbonic ...
Investigation of acetylcholinesterase and mammalian DNA topoisomerases, carbonic anhydrase inhibition profiles, and cytotoxic activity of novel bis(-aminoalkyl)phosphinic acid derivatives against human breast cancer
(Wiley, 2017-11)
The aim of this study was to evaluate biologically active novel molecules having potentials to be drugs by their antitumor properties and by activities of apoptotic caspase and topoisomerase. Following syntheses of novel ...
Synthesis of new cyclic thioureas and evaluation of their metal-chelating activity, acetylcholinesterase, butyrylcholinesterase, and carbonic anhydrase inhibition profiles
(Wiley, 2017-07)
In the presence of trifluoracetic acid (TFAA), an efficient method for the synthesis of tetra(hexa)hydropyrimidinethione-carboxylates has been used on the basis of three-component condensation of thiourea with its different ...
Synthesis of mannich bases by two different methods and evaluation of their acetylcholine esterase and carbonic anhydrase inhibitory activities
(Letters in Drug Design & Discovery, 2017)
Background: Mannich bases are an important compounds in medicinal chemistry. They have wide range of biological activities including carbonic anhydrase (CA) inhibitory and acetylcholine esterase inhibitory (AChE) activities. ...
Etkili konuşma öz yeterlik ölçeği: geçerlik ve güvenirlik çalışması
(2017)
Öğretmenlerin bildiklerini aktarmada, öğrencilerine rehberlik etmede en önemli rolü iletişim oluşturmaktadır. İletişimin temelinde ise etkili ve güzel konuşma vardır. Bu nedenle öğretmen adaylarına güzel, doğru ve etkili ...
Kelime öğretim yöntemlerinin kelime hazinesinin gelişimindeki etkisinin karşılaştırılması: meta analitik bir değerlendirme
(2017-07-29)
Eğitim araştırmalarındaki en eski alanlardan biri olan kelime öğretiminin, bireylerin anlama ve anlatma becerilerinin yanında sosyal ve iletişimsel becerilerinin de gelişimine katkı sağlayan bir etkinlik alanı olduğu kabul ...
Weierstrass representation degree and classes of the surfaces in the four dimensional Euclidean space
(Celal Bayar University, 2017)
We study two parameters families of Bour-type and Enneper-type minimal surfaces using the Weierstrass representation in the four dimensional Euclidean space. We obtain implicit algebraic equations, degree and classes of ...
Mekke kadısı Amasyalı Buhârî Şârihi Zenbillizâde Fudayl Çelebi
(Amasya Üniversitesi, 2017-12-15)
Amasya Müftüsü Zenbilli Ali Efendi'nin oğlu olan Fudayl Çelebi, 1514 İstanbul'da doğmuştur. Kânûnî Sultan Süleyman döneminin Şeyhulislam'ı olan Ebûssuûd Efendi'nin de damadıdır. Dönemin iki meşhûr âliminin ilimlerinden ...
Thermowood metodu ile ısıl işlem görmüş İsveç çamı, Sibirya çamı ve sarıçam odunlarında bazı yüzey özelliklerinin belirlenmesi
(International Advanced Researches & Engineering Congress, 2017-11-16)
In this study, it is aimed to determine the values of the color (L*, a*, b*, ΔL*, Δb*, Δa*ve ΔE*) values and
perpendicular and parallel glossiness values of define according to the ThermoWood method heat treated at 212oC ...